Palladium-catalysed direct arylation of heteroaromatics using free-NH2 iodoanilines with inhibition of amination reaction - Université de Rennes Accéder directement au contenu
Article Dans Une Revue Synthesis: Journal of Synthetic Organic Chemistry Année : 2012

Palladium-catalysed direct arylation of heteroaromatics using free-NH2 iodoanilines with inhibition of amination reaction

Résumé

The palladium-catalysed direct arylation of heteroaromatics with unprotected iodoanilines proceeds in moderate to high yields using only 1 mol% Pd(OAc)2 as the catalyst and potassium acetate as the base. No amination reaction was observed under these conditions. A wide variety of heteroarenes have been successfully employed.

Domaines

Catalyse
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Dates et versions

hal-00870547 , version 1 (07-10-2013)

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Citer

Anissa Beladhria, Kassem Beydoun, Hamed Ben Ammar, Ridha Ben Salem, Henri Doucet. Palladium-catalysed direct arylation of heteroaromatics using free-NH2 iodoanilines with inhibition of amination reaction. Synthesis: Journal of Synthetic Organic Chemistry, 2012, 44 (14), pp.2264-2276. ⟨10.1055/s-0031-1291124⟩. ⟨hal-00870547⟩
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