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Structure: Internal structure identifier : 36467
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Discovery of potent dual ligands for dopamine D4 and σ1 receptors

Nicolas Levoin , A Murthy , Vennu Narendar , Nangunoori Sampath Kumar , Pasula Aparna et al.
Bioorganic and Medicinal Chemistry, 2022, 69, pp.116851. ⟨10.1016/j.bmc.2022.116851⟩
Journal articles hal-03716651v1

Synthesis of peptidomimetics and chemo-biological tools for CD95/PLC gamma 1 interaction analysis

Ha Thanh Nguyen , Jean-Philippe Guégan , Amanda Poissonnier , Florence Jouan , Daniel Best et al.
Bioorganic and Medicinal Chemistry Letters, 2019, 29 (16), pp.2094-2099. ⟨10.1016/j.bmcl.2019.07.006⟩
Journal articles hal-02278513v1
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Structural revision of the Mcl-1 inhibitor MIM1: synthesis and biological studies on ovarian cancer cells with evaluation of designed analogues

Hippolyte Paysant , Siham Hedir , Frédéric Justaud , Louis Bastien Weiswald , Assaad Nasr El Dine et al.
Organic & Biomolecular Chemistry, 2021, 19 (41), pp.8968-8987. ⟨10.1039/d1ob01521d⟩
Journal articles hal-03414007v1
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Structure Activity Relationship Studies around DB18, a Potent and Selective Inhibitor of CLK Kinases

Dabbugoddu Brahmaiah , Anagani Kanaka Durga Bhavani , Pasula Aparna , Nangunoori Sampath Kumar , Hélène Solhi et al.
Molecules, 2022, 27 (19), pp.6149. ⟨10.3390/molecules27196149⟩
Journal articles hal-03828358v1
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Synthesis and biological studies of new piperidino-1,2,3-triazole hybrids with 3-aryl isoxazole side chains

Appala Venkata Ramana Murthy , Vennu Narendar , Nangunoori Sampath Kumar , Pasula Aparna , Anagani Kanaka Durga Bhavani et al.
Bioorganic & Medicinal Chemistry Letters, 2021, 52, pp.128390. ⟨10.1016/j.bmcl.2021.128390⟩
Journal articles hal-03414697v1
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MMP7 cleavage of amino-terminal CD95 death receptor switches signaling toward non-apoptotic pathways

Shoji F Kenji , Keerthi Kurma , Brigitte Collet , Christelle Oblet , Laure Debure et al.
Cell Death and Disease, 2022, 13 (10), pp.895. ⟨10.1038/s41419-022-05352-0⟩
Journal articles hal-03829415v1
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CD95 Structure, Aggregation and Cell Signaling

Nicolas Levoin , Mickael Jean , Patrick Legembre
Frontiers in Cell and Developmental Biology, 2020, 8, pp.314. ⟨10.3389/fcell.2020.00314⟩
Journal articles hal-02862235v1
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Synthesis and biological evaluation of FJ-809, a compound originally described as MIM1 and inhibitor of the anti-apoptotic protein Mcl-1

Frédéric Justaud , Hippolyte Paysant , Louis Bastien Weiswald , Abdelghani Jebahi , Marie Jouanne et al.
New Journal of Chemistry, 2022, 46 (19), pp.9119-9127. ⟨10.1039/D1NJ05987D⟩
Journal articles hal-03713884v1
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Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinase

Dabbugoddu Brahmaiah , Anagani Kanaka Durga Bhavani , Pasula Aparna , Nangunoori Sampath Kumar , Hélène Solhi et al.
Bioorganic and Medicinal Chemistry, 2021, 31, pp.115962. ⟨10.1016/j.bmc.2020.115962⟩
Journal articles hal-03128547v1