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cdc-like/dual-specificity tyrosine phosphorylation-regulated kinases inhibitor leucettine L41 induces mTOR-dependent autophagy: implication for Alzheimer's disease.
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Emilie Durieu
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inserm-01012086v1
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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases
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Wacothon-Karime Coulibaly
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Sibiriline, a new small chemical inhibitor of receptor-interacting protein kinase 1, prevents immune-dependent hepatitis
F. Le Cann
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C. Delehouzé
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases
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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines
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Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors
Camille Déliko Dago
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Wacothon Karime Coulibaly
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Janat A. Mamyrbekova-Bekro
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hal-01414293v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi
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William Erb
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Frédéric Lassagne
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Yury Halauko
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hal-03875302v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
M. Hedidi
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W. Erb
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G. Bentabed-Ababsa
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Floris Chevallier
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L. Picot
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hal-01381138v1
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30th Franco-Belgian conference of pharmacochemistry
Charlotte Bouckaert
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Eric Goffin
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Sebastien Dilly
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Julien Hanson
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hal-02141338v1
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6E11, a highly selective inhibitor of Receptor-Interacting Protein Kinase 1, protects cells against cold hypoxia-reoxygenation injury
C. Delehouzé
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S. Leverrier-Penna
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F. Le Cann
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A. Comte
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M. Jacquard-Fevai
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hal-01616456v1
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Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3
Killian Oukoloff
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Nicolas Coquelle
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Manuela Bartolini
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Marina Naldi
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Rémy Le Guével
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hal-02055769v1
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2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities
Nahida Mokhtari Brikci-Nigassa
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Ghenia Bentabed-Ababsa
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William Erb
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Floris Chevallier
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Laurent Picot
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hal-01774406v1
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Synthesis of new pyridazino[4,5-b]indol-4-ones and pyridazin-3(2H)-one analogs as DYRK1A inhibitors
Amélie Bruel
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Romain Bénéteau
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Mylène Chabanne
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Olivier Lozach
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hal-01086026v1
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Bioactive Metabolites from the Deep Subseafloor Fungus Oidiodendron griseum UBOCC-A-114129
Marion Navarri
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C. Jégou
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Sandrine Pottier
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hal-01518044v1
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Synthesis of New N,N'-Bis(5-arylidene-4-oxo-4,5-dihydrothiazolin-2-yl)piperazine Derivatives Under Microwave Irradiation and Preliminary Biological Evaluation.
Wacothon Karime Coulibaly
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Ludovic Paquin
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Anoubilé Bénié
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Yves-Alain Bekro
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Emilie Durieux
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inserm-00864810v1
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New 5-ylidene rhodanine derivatives based on the dispacamide A model.
Solène Guihéneuf
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Ludovic Paquin
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François Carreaux
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Emilie Durieu
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Thierry Roisnel
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hal-01017003v1
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Fused Systems Based on 2-Aminopyrimidines: Synthesis Combining Deprotolithiation-in situ Zincation with N -Arylation Reactions and Biological Properties
Madani Hedidi
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Julien Maillard
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William Erb
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Frédéric Lassagne
,
Yury S Halauko
et al.
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hal-01624382v1
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Novel optimization of valmerins (tetrahydropyrido[1,2-a]isoindolones) as potent dual CDK5/GSK3 inhibitors
Aziz Ouach
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Rajâa Boulahjar
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Christine Vala
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Stéphane Bourg
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Pascal Bonnet
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Journal articles
hal-01295635v1
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A combined experimental and theoretical study of the thermal [3+2] cycloaddition of carbonyl ylides with activated alkenes
Samira Hamza-Reguig
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Ghenia Bentabed-Ababsa
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Luis R Domingo
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Mar Ríos-Gutiérrez
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Stephanie Philippot
et al.
Journal articles
hal-01695551v2
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Novel Tetrahydropyrido[1,2-a]isoindolone Derivatives (Valmerins): Potent Cyclin-Dependent Kinase/Glycogen Synthase Kinase 3 Inhibitors with Antiproliferative Activities and Antitumor Effects in Human Tumor Xenografts
Rajâa Boulahjar
,
Aziz Ouach
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Chiurato Matteo
,
Stéphane Bourg
,
Myriam Ravache
et al.
Journal of Medicinal Chemistry, 2012, 55, pp.9589-9606
Journal articles
hal-00785213v1
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