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A practical multi-step synthesis of ethyl N-functionalized β-amino benzimidazole acrylate derivatives as promising cytotoxic agents
Christelle N'Ta Ambeu
,
Rémy Le Guével
,
Anne Corlu
,
Janat Akhanovna Mamyrbekova
,
Jean-Pierre Bazureau
et al.
Journal articles
hal-01808102v1
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Reactivity Under Microwave Irradiation of 2-amino 4H-chromene-3-carbonitrile as tool for the construction of potential bioactive derivatives
Ali Bouattour
,
Mehdi Fakhfakh
,
Houcine Ammar
,
Ludovic Paquin
,
Jean-Pierre Bazureau
et al.
3rd International Electronic Conference on Medicinal Chemistry, Nov 2022, Online, France
Conference papers
hal-03872422v1
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Comparative localization and functional activity of the main hepatobiliary transporters in HepaRG cells and primary human hepatocytes.
Pamela Bachour-El Azzi
,
Ahmad Sharanek
,
Audrey Burban
,
Ruoya Li
,
Rémy Le Guével
et al.
Journal articles
hal-01134682v1
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Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors
Camille Déliko Dago
,
Wacothon Karime Coulibaly
,
Yves-Alain Bekro
,
Janat A. Mamyrbekova-Bekro
,
Beatrice Foll-Josselin
et al.
Journal articles
hal-01414293v1
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Synthesis and biological evaluation of 3-amino-, 3-alkoxy- and 3-aryloxy-6-(hetero)arylpyridazines as potent antitumor agents
Stephane Sengmany
,
Mathilde Sitter
,
Eric Léonel
,
Erwan Le Gall
,
Gervaise Loirand
et al.
Journal articles
hal-02053836v1
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Investigation on the synthesis of new 3-[4-(arylalkoxy)phenylethyl]-2-thioxo-1,3-thiazolidin-4-ones and their biological evaluation against cancer cells
Camille Déliko Dago
,
Christelle N'Ta Ambeu
,
Wacothon Karime Coulibaly
,
Yves-Alain Békro
,
Janat A. Mamyrbekova-Bekro
et al.
Journal articles
hal-01586061v1
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Hypoxia differentially modulates the genomic stability of clinical-grade ADSCs and BM-MSCs in long-term culture
Nicolas Bigot
,
Audrey Mouche
,
Milena Preti
,
Séverine Loisel
,
Marie-Laure Renoud
et al.
Journal articles
hal-01214007v1
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Monoclonal antibodies against human translation termination factor eRF3 and their utilization for sub-cellular localization of eRF3.
Marie-Madeleine Delage
,
Stéphanie Dutertre
,
Rémy Le Guével
,
Ludmila Frolova
,
Nadia Berkova
et al.
Journal articles
inserm-00582996v1
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Inflammatory cytokines promote the retrodifferentiation of tumor-derived hepatocyte-like cells to progenitor cells.
Hélène Dubois-Pot-Schneider
,
Karim Fekir
,
Cédric Coulouarn
,
Denise Glaise
,
Caroline Aninat
et al.
Journal articles
hal-01134747v1
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Staphylococcus aureus-induced cytopathic effect on the mammalian cells
Ludmila Alekseeva
,
Rémy Le Guével
,
Lucie Rault
,
Caroline Le Marechal
,
Claire Piquet-Pellorce
et al.
4 Congress of European Microbiologists FEMS 2011, Jun 2011, Genève, Switzerland. , 2011
Conference poster
hal-02808973v1
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Direct cooperation between estrogen receptors and astrocyte-specific factors elicits high activity of the zebrafish brain aromatase gene
Arnaud Menuet
,
Elisabeth Pellegrini
,
Isabelle Anglade
,
Rémy Le Guével
,
Olivier Kah
et al.
2nd International Meeting Steroids and nervous system, February 22-26, Torino, Italy, 2003, Torino, Italy
Conference papers
hal-00107019v1
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Microwave-assisted practical synthesis of 4-imino-3-phenyl-3,4-dihydro-1H-chromeno[2,3-d]pyrimidine-2(5H)-thione derivatives and exploration of their biological activities
A. Bouattour
,
M. Fakhfakh
,
S. Abid
,
L. Paquin
,
A. Corlu
et al.
Journal articles
hal-01581215v1
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Synthesis and toxicity evaluation of hydrophobic Ionic Liquids for Volatile Organic Compounds biodegradation in a two-phase partitioning bioreactor
Alfredo Santiago Rodriguez Castillo
,
Solene Guiheneuf
,
Rémy Le Guével
,
Pierre-François Biard
,
Ludovic Paquin
et al.
Journal articles
hal-01254799v1
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Two new cyclobutane dimers from Diospyros macrocarpa
C. Thieury
,
G. Herbette
,
V. Monnier
,
N. Lebouvier
,
E. Hnawia
et al.
Journal articles
hal-01619687v1
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Expression and regulation of brain aromatase in teleost fish.
Olivier Kah
,
Arnaud Menuet
,
Elisabeth Pellegrini
,
Rémy Le Guével
,
Marie-Madeleine Guéguen
et al.
Symposium on Fish Growth and Reproduction, October 26-29, Keelung, Taiwan, 2003, Keelung, Taiwan
Conference papers
hal-00106939v1
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Structure-based design of human immuno- and constitutive proteasomes inhibitors
N. Richy
,
D. Sarraf
,
X. Maréchal
,
N. Janmamode
,
E. Genin
et al.
Journal articles
hal-01713510v1
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Structure Activity Relationship Studies around DB18, a Potent and Selective Inhibitor of CLK Kinases
Dabbugoddu Brahmaiah
,
Anagani Kanaka Durga Bhavani
,
Pasula Aparna
,
Nangunoori Sampath Kumar
,
Hélène Solhi
et al.
Journal articles
hal-03828358v1
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Prospective study directed to the synthesis of unsymmetrical linked bis-5-arylidene rhodanine derivatives via “one-pot two steps” reactions under microwave irradiation with their antitumor activity
Wacothon Karime Coulibaly
,
Ludovic Paquin
,
Anoubilé Bénie
,
Yves-Alain Békro
,
Rémy Le Guével
et al.
Journal articles
hal-01114518v1
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Biological and biophysical properties of the histone deacetylase inhibitor suberoylanilide hydroxamic Acid are affected by the presence of short alkyl groups on the phenyl ring.
Frédérik Oger
,
Aurélien Lecorgne
,
Elisa Sala
,
Vanessa Nardese
,
Florence Demay
et al.
Journal articles
hal-00462114v1
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Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3
Killian Oukoloff
,
Nicolas Coquelle
,
Manuela Bartolini
,
Marina Naldi
,
Rémy Le Guével
et al.
Journal articles
hal-02055769v1
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Identification of small molecule regulators of the nuclear receptor HNF4alpha based on naphthofuran scaffolds.
Rémy Le Guével
,
Frédérik Oger
,
Aurélien Lecorgne
,
Zuzana Dudasova
,
Soizic Chevance
et al.
Journal articles
istex
hal-00422061v1
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Toxicologie predictive: les voies du futur
Ph Detilleux
,
L Vallier
,
C Legallais
,
E Leclerc
,
M Prot J
et al.
Congrès de la SPTC - Société de Pharmaco-Toxicologie Cellulaire, May 2010, Paris, France
Conference papers
hal-01122677v1
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The novel antibacterial compound walrycin A induces human PXR transcriptional activity.
Alexandre Berthier
,
Frédérik Oger
,
Céline Gheeraert
,
Abdel Boulahtouf
,
Rémy Le Guével
et al.
Journal articles
inserm-00672104v1
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Synthesis and biological studies of new quinazolines with ether functions in position 2
D. Brahmaiah
,
A.K.D. Bhavani
,
P. Aparna
,
N.S. Kumar
,
H. Solhi
et al.
Journal articles
hal-02161844v1
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Electrochemical synthesis and characterisation of alternating tripyridyl-dipyrrole molecular strands with multiple nitrogen-based donor-acceptor binding sites.
Alexandra Tabatchnik-Rebillon
,
Christophe Aubé
,
Hicham Bakkali
,
Thierry Delaunay
,
Gabriel Thia Manh
et al.
Journal articles
istex
hal-00742561v1
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Mechanisms of action and structure-activity relationships of cytotoxic flavokawain derivatives
Charlotte Thieury
,
Nicolas Lebouvier
,
Rémy Le Guével
,
Yann Barguil
,
Gaëtan Herbette
et al.
Journal articles
hal-01485126v1
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Inactivation of the Nuclear Orphan Receptor COUP-TFII by Small Chemicals
Rémy Le Guével
,
Frederik Oger
,
Celia P. Martinez-Jimenez
,
Maud Bizot
,
Celine Gheeraert
et al.
Journal articles
hal-01497231v1
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Inactivation of AMPK in human granulosa cells
Pascal Froment
,
Charlène Rouillon
,
Joëlle Dupont
,
I Plotton
,
Rémy Le Guével
et al.
50. Annual meeting of the Society for the Study of Reproduction SSR, 2017, washington, United States. , 2017
Conference poster
hal-02787865v1
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Synthesis of New N,N'-Bis(5-arylidene-4-oxo-4,5-dihydrothiazolin-2-yl)piperazine Derivatives Under Microwave Irradiation and Preliminary Biological Evaluation.
Wacothon Karime Coulibaly
,
Ludovic Paquin
,
Anoubilé Bénié
,
Yves-Alain Bekro
,
Emilie Durieux
et al.
Journal articles
inserm-00864810v1
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Distribution of aromatase mRNA and protein in the brain and pituitary of female rainbow trout: Comparison with estrogen receptor alpha.
Arnaud Menuet
,
Isabelle Anglade
,
Rémy Le Guével
,
Elisabeth Pellegrini
,
Farzad Pakdel
et al.
Journal articles
istex
hal-00295588v1
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