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Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors
Camille Déliko Dago
,
Wacothon Karime Coulibaly
,
Yves-Alain Bekro
,
Janat A. Mamyrbekova-Bekro
,
Beatrice Foll-Josselin
et al.
Journal articles
hal-01414293v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi
,
Julien Maillard
,
William Erb
,
Frédéric Lassagne
,
Yury Halauko
et al.
Journal articles
hal-03875302v1
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30th Franco-Belgian conference of pharmacochemistry
Charlotte Bouckaert
,
Eric Goffin
,
Sebastien Dilly
,
Julien Hanson
,
Lionel Pochet
et al.
Journal articles
hal-02141338v1
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Reactivity Under Microwave Irradiation of 2-amino 4H-chromene-3-carbonitrile as tool for the construction of potential bioactive derivatives
Ali Bouattour
,
Mehdi Fakhfakh
,
Houcine Ammar
,
Ludovic Paquin
,
Jean-Pierre Bazureau
et al.
3rd International Electronic Conference on Medicinal Chemistry, Nov 2022, Online, France
Conference papers
hal-03872422v1
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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines
Frédéric Lassagne
,
Timothy Langlais
,
Elsa Caytan
,
Emmanuelle Limanton
,
Ludovic Paquin
et al.
Journal articles
hal-03867783v1
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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases
Camille Déliko Dago
,
Christelle Ambeu
,
Wacothon-Karime Coulibaly
,
Yves-Alain Békro
,
Janat Mamyrbékova
et al.
Journal articles
hal-01187427v1
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Structure Activity Relationship Studies around DB18, a Potent and Selective Inhibitor of CLK Kinases
Dabbugoddu Brahmaiah
,
Anagani Kanaka Durga Bhavani
,
Pasula Aparna
,
Nangunoori Sampath Kumar
,
Hélène Solhi
et al.
Journal articles
hal-03828358v1
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2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities
Nahida Mokhtari Brikci-Nigassa
,
Ghenia Bentabed-Ababsa
,
William Erb
,
Floris Chevallier
,
Laurent Picot
et al.
Journal articles
hal-01774406v1
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Design, biological evaluation and X-ray crystallography of nanomolar multifunctional ligands targeting simultaneously acetylcholinesterase and glycogen synthase kinase-3
Killian Oukoloff
,
Nicolas Coquelle
,
Manuela Bartolini
,
Marina Naldi
,
Rémy Le Guével
et al.
Journal articles
hal-02055769v1
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Bioactive Metabolites from the Deep Subseafloor Fungus Oidiodendron griseum UBOCC-A-114129
Marion Navarri
,
C. Jégou
,
Arnaud Bondon
,
Sandrine Pottier
,
Stéphane Bach
et al.
Journal articles
hal-01518044v1
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Fused Systems Based on 2-Aminopyrimidines: Synthesis Combining Deprotolithiation-in situ Zincation with N -Arylation Reactions and Biological Properties
Madani Hedidi
,
Julien Maillard
,
William Erb
,
Frédéric Lassagne
,
Yury S Halauko
et al.
Journal articles
hal-01624382v1
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Novel optimization of valmerins (tetrahydropyrido[1,2-a]isoindolones) as potent dual CDK5/GSK3 inhibitors
Aziz Ouach
,
Rajâa Boulahjar
,
Christine Vala
,
Stéphane Bourg
,
Pascal Bonnet
et al.
Journal articles
hal-01295635v1
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A combined experimental and theoretical study of the thermal [3+2] cycloaddition of carbonyl ylides with activated alkenes
Samira Hamza-Reguig
,
Ghenia Bentabed-Ababsa
,
Luis R Domingo
,
Mar Ríos-Gutiérrez
,
Stephanie Philippot
et al.
Journal articles
hal-01695551v2
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Functionalization of 9-thioxanthone at the 1-position: From arylamino derivatives to [1]benzo(thio)pyrano[4,3,2-de]benzothieno[2,3-b]quinolines of biological interest
Nahida Mokhtari Brikci-Nigassa
,
Lionel Nauton
,
Pascale Moreau
,
Olivier Mongin
,
Raphael E Duval
et al.
Journal articles
hal-02404054v1
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Discovery of DB18, a potent inhibitor of CLK kinases with a high selectivity against DYRK1A kinase
Dabbugoddu Brahmaiah
,
Anagani Kanaka Durga Bhavani
,
Pasula Aparna
,
Nangunoori Sampath Kumar
,
Hélène Solhi
et al.
Journal articles
hal-03128547v1
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From simple quinoxalines to potent oxazolo[5,4-f]quinoxaline inhibitors of glycogen-synthase kinase 3 (GSK3)
Frédéric Lassagne
,
Camille Duguépéroux
,
Carlos Roca
,
Concepción Pérez
,
Ana Martínez
et al.
Journal articles
hal-02396922v1
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Synthesis of New 2-Phenylamino-4H-chromene-3-carbonitrile Derivatives and Their Effects on Tumor Cell Lines and against Protein Kinases
Ali Bouattour
,
Mehdi Fakhfakh
,
Souhir Abid
,
Ludovic Paquin
,
Rémy Le Guével
et al.
Journal articles
hal-03869130v2
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Azine and Diazine Functionalization Using 2,2,6,6-Tetramethylpiperidino-Based Lithium–Metal Combinations: Application to the Synthesis of 5,9-Disubstituted Pyrido[3′,2′:4,5]pyrrolo[1,2-c] pyrimidines
Nada Marquise
,
Tan Tai Nguyen
,
Floris Chevallier
,
Laurent Picot
,
Valérie Thiéry
et al.
Journal articles
hal-01248092v1
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