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Encapsulation of (E)-N’-(1-(7-(diethylamino)-2-oxo-2H-chromen-3 yl)ethylidene)benzohydrazide (7-diEAHC) in β-cyclodextrins: Optimized synthesis of 7-diEACH and in silico ADME profiling, physical stability, antioxidant properties of encapsulated 7-diEAHC and bioavailability in rats
E. Khdhiri
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S Abid
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K. Athmouni
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M. Abid
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H. Ayadi
et al.
Journal articles
hal-03975255v1
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Sample preparation for an optimized extraction of localized metabolites in lichens: Application to Pseudevernia furfuracea
Sarah Komaty
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Marine Letertre
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Huyen Duong Dang
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Harald Jungnickel
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Peter Laux
et al.
Journal articles
hal-01254800v1
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A Practical Approach to New (5Z) 2-Alkylthio-5-arylmethylene- 1-methyl-1,5-dihydro-4H-imidazol-4-one Derivatives
Khadidja Bourahla
,
Ludovic Paquin
,
Olivier Lozach
,
Laurent Meijer
,
François Carreaux
et al.
Journal articles
hal-00870301v1
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Ionic liquid-phase organic synthesis (IoLiPOS) methodology applied to cross aldol reaction
Halima Hakkou
,
Daniel Carrié
,
Ludovic Paquin
,
Jean-Pierre Bazureau
Journal articles
istex
hal-00869914v1
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Microwave synthesis of new 3-(3-aminopropyl)-5-arylidene-2-thioxo-1,3-thiazolidine-4-ones as potential Ser/Thr protein kinase inhibitors
Camille Déliko Dago
,
Wacothon Karime Coulibaly
,
Yves-Alain Bekro
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Janat A. Mamyrbekova-Bekro
,
Beatrice Foll-Josselin
et al.
Journal articles
hal-01414293v1
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Evolution of DMSP (dimethylsulfoniopropionate) biosynthesis pathway: Origin and phylogenetic distribution in polyploid Spartina (Poaceae, Chloridoideae)
Hélène Rousseau
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Mathieu Rousseau-Gueutin
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Xavier Dauvergne
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Julien Boutte
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Gaëlle Simon
et al.
Journal articles
hal-01579439v1
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Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B.
Tania Tahtouh
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Jonathan M. Elkins
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Panagis Filippakopoulos
,
Meera Soundararajan
,
Guillaume Burgy
et al.
Journal articles
hal-00870472v1
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Investigation on the synthesis of new 3-[4-(arylalkoxy)phenylethyl]-2-thioxo-1,3-thiazolidin-4-ones and their biological evaluation against cancer cells
Camille Déliko Dago
,
Christelle N'Ta Ambeu
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Wacothon Karime Coulibaly
,
Yves-Alain Békro
,
Janat A. Mamyrbekova-Bekro
et al.
Journal articles
hal-01586061v1
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Method for synthesizing polyesters in an acidic ionic liquid medium
Alain Fradet
,
Hervé Lefebvre
,
Jean-Pierre Bazureau
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Ludovic Paquin
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Daniel Carrié
et al.
France, Patent n° : WO2011012814 A1. 2011
Patents
hal-00873181v1
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Synthesis and preliminary biological evaluation of new derivatives of the marine alkaloid leucettamine B as kinase inhibitors.
Mansour Debdab
,
Stéven Renault
,
Olivier Lozach
,
Laurent Meijer
,
Ludovic Paquin
et al.
Journal articles
istex
hal-00869769v1
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Synthesis of 3,5-disubstituted 1,2,4-oxadiazoles using ionic liquid-phase organic synthesis (IoLiPOS) methodology
Laetitia Duchet
,
Jean-Christophe Legeay
,
Daniel Carrié
,
Ludovic Paquin
,
Jean-Jacques Vanden
et al.
Journal articles
istex
hal-00869781v1
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The Franco-Brazilian network on natural products (FB2NP): a new network promoting cooperation and exchanges in natural products research
Jackson Almeida
,
Raphaël Grougnet
,
Lucindo Quintans
,
Marc Feuilloley
,
Thomas Robert
et al.
Journal articles
hal-03592226v1
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N-Boc and N-CBz Ethyl Oxamates: New Gabriel Reagents
Fabienne Berrée
,
Jean-Pierre Bazureau
,
Gwendal Michelot
,
Maurice Le Cone
Journal articles
hal-03985910v1
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Studies of the Chemical Reactivity of a Series of Rhodanine Derivatives by Approaches to Quantum Chemistry
Wacothon Karime Coulibaly
,
Jean Stéphane N’dri
,
Mamadou Guy-Richard Koné
,
Camille Déliko Dago
,
Christelle N’ta Ambeu
et al.
Journal articles
hal-02572308v1
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Microwave Assisted Organic Synthesis (MAOS) of New Dispacamide A Derivatives Bearing a Thiazolinone Platform, Biological Assays on Inhibition of Protein Kinases and Cell Effects
Solene Guiheneuf
,
Ludovic Paquin
,
Francois Carreaux
,
Emilie Durieu
,
Helene Benedetti
et al.
Journal articles
hal-01114583v1
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30th Franco-Belgian conference of pharmacochemistry
Charlotte Bouckaert
,
Eric Goffin
,
Sebastien Dilly
,
Julien Hanson
,
Lionel Pochet
et al.
Journal articles
hal-02141338v1
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1,3-dipolar cycloadditions of aldehydes or Imines with carbonyl ylides generated from epoxides: Classical heating and microwave irradiation
Ghenia Bentabed-Ababsa
,
Mustapha Rahmouni
,
Florence Mongin
,
Aicha Derdour
,
Jack. Hamelin
et al.
Journal articles
hal-00781884v1
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Practical approach to N-benzyl derivatives of 2-amino-8-methoxy-4H-chromene-3-carbonitrile by reductive amination: Exploration of their effects against protein kinases and in silico ADME profiling
Marwa Dhiabi
,
Ali Bouattour
,
Mehdi Fakhfakh
,
Souhir Abid
,
Ludovic Paquin
et al.
Journal articles
hal-03867314v1
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Leucettines, a class of potent inhibitors of cdc2-like kinases and dual specificity, tyrosine phosphorylation regulated kinases derived from the marine sponge leucettamine B: modulation of alternative pre-RNA splicing.
Mansour Debdab
,
François Carreaux
,
Steven Renault
,
Meera Soundararajan
,
Oleg Fedorov
et al.
Journal articles
hal-00870007v1
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An efficient approach to dispacamide A and its derivatives.
Solène Guihéneuf
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Ludovic Paquin
,
François Carreaux
,
Emilie Durieu
,
Laurent Meijer
et al.
Journal articles
hal-00870469v1
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(E)-N'-(1-(3-oxo-3H-benzo[f]chromen-2-yl)ethylidene)benzohydrazide protecting rat heart tissues from isoproterenol toxicity: Evidence from in vitro and in vivo tests
Khdhiri Emna
,
Kais Mnafgui
,
Lakhdar Ghazouani
,
Anouar Feriani
,
Raouf Hajji
et al.
Journal articles
hal-02635141v1
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cdc-like/dual-specificity tyrosine phosphorylation-regulated kinases inhibitor leucettine L41 induces mTOR-dependent autophagy: implication for Alzheimer's disease.
Xavier Fant
,
Emilie Durieu
,
Gaëtan Chicanne
,
Bernard Payrastre
,
Diego Sbrissa
et al.
Journal articles
inserm-01012086v1
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Reactivity Under Microwave Irradiation of 2-amino 4H-chromene-3-carbonitrile as tool for the construction of potential bioactive derivatives
Ali Bouattour
,
Mehdi Fakhfakh
,
Houcine Ammar
,
Ludovic Paquin
,
Jean-Pierre Bazureau
et al.
3rd International Electronic Conference on Medicinal Chemistry, Nov 2022, Online, France
Conference papers
hal-03872422v1
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Structure-Activity Relationship in the Leucettine Family of Kinase Inhibitors
Tania Tahtouh
,
Emilie Durieu
,
Benoit Villiers
,
Celine Bruyere
,
Thu Lan Nguyen
et al.
Journal articles
hal-03512536v1
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases
Nadège Loaëc
,
Eletta Attanasio
,
Benoît Villiers
,
Emilie Durieu
,
Tania Tahtouh
et al.
Journal articles
hal-01640115v1
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A practical multi-step synthesis of ethyl N-functionalized β-amino benzimidazole acrylate derivatives as promising cytotoxic agents
Christelle N'Ta Ambeu
,
Rémy Le Guével
,
Anne Corlu
,
Janat Akhanovna Mamyrbekova
,
Jean-Pierre Bazureau
et al.
Journal articles
hal-01808102v1
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Leucettine L41, a DYRK1A-preferential DYRKs/CLKs inhibitor, prevents memory impairments and neurotoxicity induced by oligomeric Aβ25-35 peptide administration in mice.
Gaëlle Naert
,
Valentine Ferré
,
Johann Meunier
,
Emeline Keller
,
Susanna Malmstrom
et al.
Journal articles
hal-01146496v1
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Synthetic Development of New 3-(4-Arylmethylamino)butyl-5-arylidene-rhodanines under Microwave Irradiation and Their Effects on Tumor Cell Lines and against Protein Kinases
Camille Déliko Dago
,
Christelle Ambeu
,
Wacothon-Karime Coulibaly
,
Yves-Alain Békro
,
Janat Mamyrbékova
et al.
Journal articles
hal-01187427v1
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Anti-proliferative Activity Study on 5-Arylidene Rhodanine Derivatives Using Density Functional Theory (DFT) and Quantitative Structure Activity Relationship (QSAR)
Wacothon Coulibaly
,
Affi Sopi
,
James Titah
,
Guy-Richard Koné
,
Affoué Estelle
et al.
Journal articles
hal-03988161v1
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Correction of cognitive deficits in mouse models of Down syndrome by a pharmacological inhibitor of DYRK1A
Thu Lan Nguyen
,
Arnaud Duchon
,
Antigoni Manousopoulou
,
Nadège Loaëc
,
Benoît Villiers
et al.
Journal articles
hal-01862465v1
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