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[3,3]-Sigmatropic Rearrangement of Boronated Allylcyanates: A New Route to α-Aminoboronate Derivatives and Trisubstituted Tetrahydrofurans
Sabrina Touchet
,
Aurélie Macé
,
Thierry Roisnel
,
François Carreaux
,
Alexandre Bouillon
et al.
Organic Letters, 2013, 15 (11), pp.2712-2715
Journal articles
hal-02029934v1
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Boron- and silicon-substituted [3]-1-heterodendralenes as versatile building blocks for the rapid construction of polycyclic architectures.
Fabien Tripoteau
,
Tristan Verdelet
,
Alain Hercouet
,
François Carreaux
,
Bertrand Carboni
et al.
Journal articles
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hal-00869895v1
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An efficient approach to dispacamide A and its derivatives.
Solène Guihéneuf
,
Ludovic Paquin
,
François Carreaux
,
Emilie Durieu
,
Laurent Meijer
et al.
Journal articles
hal-00870469v1
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[3,3]-Sigmatropic Rearrangement/Allylboration/Cyclization Sequence: Enantioenriched Seven-Membered-Ring Carbamates and Ring Contraction to Pyrrolidines
Aurélie Macé
,
Sabrina Touchet
,
Patricia Andres
,
Fernando Cossío
,
Vincent Dorcet
et al.
Journal articles
istex
hal-01240655v1
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cdc-like/dual-specificity tyrosine phosphorylation-regulated kinases inhibitor leucettine L41 induces mTOR-dependent autophagy: implication for Alzheimer's disease.
Xavier Fant
,
Emilie Durieu
,
Gaëtan Chicanne
,
Bernard Payrastre
,
Diego Sbrissa
et al.
Journal articles
inserm-01012086v1
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Leucettines, a class of potent inhibitors of cdc2-like kinases and dual specificity, tyrosine phosphorylation regulated kinases derived from the marine sponge leucettamine B: modulation of alternative pre-RNA splicing.
Mansour Debdab
,
François Carreaux
,
Steven Renault
,
Meera Soundararajan
,
Oleg Fedorov
et al.
Journal articles
hal-00870007v1
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Leucettine L41, a DYRK1A-preferential DYRKs/CLKs inhibitor, prevents memory impairments and neurotoxicity induced by oligomeric Aβ25-35 peptide administration in mice.
Gaëlle Naert
,
Valentine Ferré
,
Johann Meunier
,
Emeline Keller
,
Susanna Malmstrom
et al.
Journal articles
hal-01146496v1
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Alkenylboron Cross-Coupling
Bertrand Carboni
,
François Carreaux
Mats Larhed, John P. Wolfe, G. Molander. Science of Synthesis, Georg Thieme Verlag, pp.265-322, 2012
Book sections
hal-00873122v1
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Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases
Nadège Loaëc
,
Eletta Attanasio
,
Benoît Villiers
,
Emilie Durieu
,
Tania Tahtouh
et al.
Journal articles
hal-01640115v1
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Microwave-Assisted 1,3-Dioxa-[3,3]-Sigmatropic Rearrangement of Substituted Allylic Carbamates: Application to the Synthesis of Novel 1,3-Oxazine-2,4-dione Derivatives
Samar Bou Zeid
,
Samar Eid
,
Fadia Najjar
,
Aurélie Macé
,
Ivan Rivilla
et al.
Journal articles
hal-03464791v1
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Structural and molecular bases to IRE1 activity modulation
Timothy Langlais
,
Diana Pelizzari-Raymundo
,
Sayyed Jalil Mahdizadeh
,
Nicolas Gouault
,
François Carreaux
et al.
Journal articles
hal-03331317v1
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Structure-Activity Relationship in the Leucettine Family of Kinase Inhibitors
Tania Tahtouh
,
Emilie Durieu
,
Benoit Villiers
,
Celine Bruyere
,
Thu Lan Nguyen
et al.
Journal articles
hal-03512536v1
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BINOL derivatives-catalysed enantioselective allylboration of isatins: application to the synthesis of (R)-chimonamidine
Julien Braire
,
Vincent Dorcet
,
Joëlle Vidal
,
Claudia Lalli
,
François Carreaux
et al.
Journal articles
hal-02928635v1
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Synthesis of alkenyl boronates from allyl-substituted aromatics using an olefin cross-metathesis protocol.
Rémy Hemelaere
,
François Carreaux
,
Bertrand Carboni
Journal articles
hal-00861076v1
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A Diastereoselective Route to trans-2-Aryl-2,3-dihydrobenzofurans through Sequential Cross-Metathesis/Isomerization/Allylboration Reactions: Synthesis of Bioactive Neolignans
Rémy Hemelaere
,
François Carreaux
,
Bertrand Carboni
Journal articles
istex
hal-01138641v1
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Pentamethylcyclopentadienyl ruthenium: an efficient catalyst for the redox isomerization of functionalized allylic alcohols into carbonyl compounds
Asmae Bouziane
,
Bertrand Carboni
,
Christian Bruneau
,
François Carreaux
,
Jean-Luc Renaud
et al.
Tetrahedron, 2008, 64, pp.11745-11750
Journal articles
hal-00356814v1
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Solid-phase reactions of resin-supported boronic acids
François Carreaux
,
Bertrand Carboni
,
Hervé Deleuze
,
Christelle Pourbaix-L'Ebraly
Book sections
hal-00873126v1
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A Practical Approach to New (5Z) 2-Alkylthio-5-arylmethylene- 1-methyl-1,5-dihydro-4H-imidazol-4-one Derivatives
Khadidja Bourahla
,
Ludovic Paquin
,
Olivier Lozach
,
Laurent Meijer
,
François Carreaux
et al.
Journal articles
hal-00870301v1
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Iridium-Catalyzed Allylic Amination Route to α-Aminoboronates: Illustration of the Decisive Role of Boron Substituents.
Sabrina Touchet
,
François Carreaux
,
Gary A. Molander
,
Bertrand Carboni
,
Alexandre Bouillon
et al.
Journal articles
hal-00869890v1
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A Practical Access to Novel 2-Amino-5-arylidene-thiazol-4-ones via Sulfur/nitrogen Displacement under Solvent-free Microwave Irradiations.
Khadidja Bourahlaa
,
Aicha Derdour
,
Mustapha Rahmouni
,
François Carreaux
,
J.P. Bazureau
et al.
Tetrahedron Letters, 2007, pp.5785-5789
Journal articles
hal-00410745v1
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Synthetic alkyl-ether-lipid promotes TRPV2 channel trafficking trough PI3K/Akt-girdin axis in cancer cells and increases mammary tumour volume
Maxime Guéguinou
,
Romain Felix
,
Séverine Marionneau-Lambot
,
Thibauld Oullier
,
Aubin Penna
et al.
Journal articles
hal-03278876v1
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Ruthenium-Catalyzed Synthesis of Allylic Alcohols: Boronic Acid as a Hydroxide Source
Asmae Bouziane
,
Marion Helou
,
Bertrand Carboni
,
François Carreaux
,
Bernard Demerseman
et al.
Chemistry, Eur., 2008, pp.5630-5637
Journal articles
hal-00356801v1
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Synthesis and preliminary biological evaluation of new derivatives of the marine alkaloid leucettamine B as kinase inhibitors.
Mansour Debdab
,
Stéven Renault
,
Olivier Lozach
,
Laurent Meijer
,
Ludovic Paquin
et al.
Journal articles
istex
hal-00869769v1
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Aminoboronic acids and esters: from synthetic challenges to the discovery of unique classes of enzyme inhibitors.
Sabrina Touchet
,
François Carreaux
,
Bertrand Carboni
,
Alexandre Bouillon
,
Jean-Luc Boucher
et al.
Journal articles
hal-00869909v1
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Dérivés d'imidazolones, procédé de préparation et applications biologiques.
J.P. Bazureau
,
François Carreaux
,
Stéven Renault
,
Laurent Meijer
,
Olivier Lozach
et al.
Patent n° : FR 291 9608 (A1). 2009
Patents
hal-00411458v1
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Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B.
Tania Tahtouh
,
Jonathan M. Elkins
,
Panagis Filippakopoulos
,
Meera Soundararajan
,
Guillaume Burgy
et al.
Journal articles
hal-00870472v1
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(E)-Α-Substituted Γ-Alkoxyallylboronic Esters as New Reagents: Synthesis and Reactivity toward Aldehydes.
Françoise Possémé
,
Michael Deligny
,
François Carreaux
,
Bertrand Carboni
Journal of Organic Chemistry, 2008, 72, pp.984-989
Journal articles
hal-00356454v1
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An expeditious, environment-friendly, and microwave-assisted synthesis of 5-isatinylidenerhodanine derivatives
Abdelmounaim Safer
,
Mustapha Rahmouni
,
François Carreaux
,
Ludovic Paquin
,
Olivier Lozach
et al.
Journal articles
hal-00869920v1
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Iridium-Catalyzed Allylic Amination Route to α-Aminoboronates: Illustration of the Decisive Role of Boron Substituents
Sabrina Touchet
,
François Carreaux
,
Gary Molander
,
Bertrand Carboni
,
Alexandre Bouillon
et al.
Advanced Synthesis and Catalysis, 2011, 353 (18), pp.3391-3396
Journal articles
hal-02029761v1
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Inhibition of DYRK1A proteolysis modifies its kinase specificity and rescues Alzheimer phenotype in APP/PS1 mice
Benoit Souchet
,
Mickael Audrain
,
Jean Marie Billard
,
Julien Dairou
,
Romain Fol
et al.
Journal articles
hal-02324924v1
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