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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines
Frédéric Lassagne
,
Timothy Langlais
,
Elsa Caytan
,
Emmanuelle Limanton
,
Ludovic Paquin
et al.
Journal articles
hal-03867783v1
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Thiazolo[5,4- f ]quinoxalines, Oxazolo[5,4- f ]quinoxalines and Pyrazino[ b,e ]isatins: Synthesis from 6-Aminoquinoxalines and Properties
Frédéric Lassagne
,
Joshua M. Sims
,
William Erb
,
Olivier Mongin
,
Nicolas Richy
et al.
Journal articles
hal-03269555v1
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Deproto-metallation using mixed lithium-zinc and lithium-copper bases and computed CH acidity of 2-substituted quinolines
Nada Marquise
,
Guillaume Bretel
,
Frédéric Lassagne
,
Floris Chevallier
,
Thierry Roisnel
et al.
Journal articles
hal-01002410v1
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Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi
,
Julien Maillard
,
William Erb
,
Frédéric Lassagne
,
Yury Halauko
et al.
Journal articles
hal-03875302v1
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Functionalization of pyridyl ketones using deprotolithiation-in situ zincation
Madani Hedidi
,
William Erb
,
Frédéric Lassagne
,
Yury S. Halauko
,
Oleg A. Ivashkevich
et al.
Journal articles
hal-01357392v1
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Oxazolo[5,4-f]quinoxaline-type selective inhibitors of glycogen synthase kinase-3α (GSK-3α): Development and impact on temozolomide treatment of glioblastoma cells
Mohamed Hasyeoui
,
Frédéric Lassagne
,
William Erb
,
Manal Nael
,
Khaled Elokely
et al.
Journal articles
hal-04059446v1
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Aromatic Iodides: Synthesis and Conversion to Heterocycles
Florence Mongin
,
William Erb
,
Frédéric Lassagne
Journal articles
hal-04059384v1
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Deprotonative Metalation of Methoxy-Substituted Arenes Using Lithium 2,2,6,6-Tetramethylpiperidide Experimental and Computational Study
Gaku Akimoto
,
Mai Otsuka
,
Ryo Takita
,
Masanobu Uchiyama
,
Madani Hedidi
et al.
Journal articles
hal-01935364v1
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Copper- and Cobalt-Catalyzed Syntheses of Thiophene-Based Tertiary Amines
Salima Bouarfa
,
Simon Graβl
,
Maria Ivanova
,
Timothy Langlais
,
Ghenia Bentabed-Ababsa
et al.
Journal articles
hal-02177982v1
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Direct metallation of thienopyrimidines using a mixed lithium-cadmium base and antitumor activity of functionalized derivatives
Katia Snégaroff
,
Frédéric Lassagne
,
Ghenia Bentabed-Ababsa
,
Nassar Ekhlass
,
Ely Sidaty Cheikh Sid
et al.
Journal articles
hal-00785054v1
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A Combined Experimental and Theoretical Study of the Ammonium Bifluoride Catalyzed Regioselective Synthesis of Quinoxalines and Pyrido[2,3-b]pyrazines
Frédéric Lassagne
,
Floris Chevallier
,
Thierry Roisnel
,
Vincent Dorcet
,
Florence Mongin
et al.
Journal articles
hal-01248104v1
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Fused Systems Based on 2-Aminopyrimidines: Synthesis Combining Deprotolithiation-in situ Zincation with N -Arylation Reactions and Biological Properties
Madani Hedidi
,
Julien Maillard
,
William Erb
,
Frédéric Lassagne
,
Yury S Halauko
et al.
Journal articles
hal-01624382v1
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A convenient synthesis of 3- and 5-amino-1H-pyrazoles via 3(5)-amino-4-(ethylsulfinyl)-1H-pyrazole desulfinylation
Frédéric Lassagne
,
Katia Snégaroff
,
Thierry Roisnel
,
Ekhlass Nassar
,
Florence Mongin
et al.
Journal articles
istex
hal-00736464v1
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From simple quinoxalines to potent oxazolo[5,4-f]quinoxaline inhibitors of glycogen-synthase kinase 3 (GSK3)
Frédéric Lassagne
,
Camille Duguépéroux
,
Carlos Roca
,
Concepción Pérez
,
Ana Martínez
et al.
Journal articles
hal-02396922v1
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Deproto-metallation and computed CH acidity of 2-aryl-1,2,3-triazoles.
Floris Chevallier
,
Thomas Blin
,
Elisabeth Nagaradja
,
Frédéric Lassagne
,
Thierry Roisnel
et al.
Journal articles
hal-01053777v1
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