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authFullName_s : Frédéric Lassagne
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From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines

Frédéric Lassagne , Timothy Langlais , Elsa Caytan , Emmanuelle Limanton , Ludovic Paquin et al.
Molecules, 2018, 23 (11), pp.2961. ⟨10.3390/molecules23112961⟩
Journal articles hal-03867783v1
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Thiazolo[5,4- f ]quinoxalines, Oxazolo[5,4- f ]quinoxalines and Pyrazino[ b,e ]isatins: Synthesis from 6-Aminoquinoxalines and Properties

Frédéric Lassagne , Joshua M. Sims , William Erb , Olivier Mongin , Nicolas Richy et al.
European Journal of Organic Chemistry, 2021, 2021 (19), pp.2756-2763. ⟨10.1002/ejoc.202100362⟩
Journal articles hal-03269555v1
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Deproto-metallation using mixed lithium-zinc and lithium-copper bases and computed CH acidity of 2-substituted quinolines

Nada Marquise , Guillaume Bretel , Frédéric Lassagne , Floris Chevallier , Thierry Roisnel et al.
RSC Advances, 2014, 4 (38), pp.19602. ⟨10.1039/c4ra02583k⟩
Journal articles hal-01002410v1

Synthesis of N-pyridyl azoles using a deprotometalation-iodolysis-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells

Madani Hedidi , Julien Maillard , William Erb , Frédéric Lassagne , Yury Halauko et al.
Tetrahedron, 2016, 72 (39), pp.6467 - 6476. ⟨10.1016/j.tet.2016.08.056⟩
Journal articles hal-03875302v1
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Functionalization of pyridyl ketones using deprotolithiation-in situ zincation

Madani Hedidi , William Erb , Frédéric Lassagne , Yury S. Halauko , Oleg A. Ivashkevich et al.
RSC Advances, 2016, 6 (68), pp.63185--63189. ⟨10.1039/c6ra11370b⟩
Journal articles hal-01357392v1
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Oxazolo[5,4-f]quinoxaline-type selective inhibitors of glycogen synthase kinase-3α (GSK-3α): Development and impact on temozolomide treatment of glioblastoma cells

Mohamed Hasyeoui , Frédéric Lassagne , William Erb , Manal Nael , Khaled Elokely et al.
Bioorganic Chemistry, 2023, 134, pp.106456. ⟨10.1016/j.bioorg.2023.106456⟩
Journal articles hal-04059446v1
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Aromatic Iodides: Synthesis and Conversion to Heterocycles

Florence Mongin , William Erb , Frédéric Lassagne
Chemistry Proceedings, 2022, 12, pp.20. ⟨10.3390/ecsoc-26-13641⟩
Journal articles hal-04059384v1
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Deprotonative Metalation of Methoxy-Substituted Arenes Using Lithium 2,2,6,6-Tetramethylpiperidide Experimental and Computational Study

Gaku Akimoto , Mai Otsuka , Ryo Takita , Masanobu Uchiyama , Madani Hedidi et al.
Journal of Organic Chemistry, 2018, 83 (21), pp.13498-13506. ⟨10.1021/acs.joc.8b02397⟩
Journal articles hal-01935364v1
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Copper- and Cobalt-Catalyzed Syntheses of Thiophene-Based Tertiary Amines

Salima Bouarfa , Simon Graβl , Maria Ivanova , Timothy Langlais , Ghenia Bentabed-Ababsa et al.
European Journal of Organic Chemistry, 2019, 2019 (20), pp.3244-3258. ⟨10.1002/ejoc.201900276⟩
Journal articles hal-02177982v1
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Direct metallation of thienopyrimidines using a mixed lithium-cadmium base and antitumor activity of functionalized derivatives

Katia Snégaroff , Frédéric Lassagne , Ghenia Bentabed-Ababsa , Nassar Ekhlass , Ely Sidaty Cheikh Sid et al.
Organic & Biomolecular Chemistry, 2009, 7 (22), pp.4782-4788. ⟨10.1039/B915274A⟩
Journal articles hal-00785054v1
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A Combined Experimental and Theoretical Study of the Ammonium Bifluoride Catalyzed Regioselective Synthesis of Quinoxalines and Pyrido[2,3-b]pyrazines

Frédéric Lassagne , Floris Chevallier , Thierry Roisnel , Vincent Dorcet , Florence Mongin et al.
Synthesis: Journal of Synthetic Organic Chemistry, 2015, 47 (17), pp.2680-2689. ⟨10.1055/s-0034-1380678⟩
Journal articles hal-01248104v1
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Fused Systems Based on 2-Aminopyrimidines: Synthesis Combining Deprotolithiation-in situ Zincation with N -Arylation Reactions and Biological Properties

Madani Hedidi , Julien Maillard , William Erb , Frédéric Lassagne , Yury S Halauko et al.
European Journal of Organic Chemistry, 2017, 2017 (39), pp.5903-5915. ⟨10.1002/ejoc.201701004⟩
Journal articles hal-01624382v1

A convenient synthesis of 3- and 5-amino-1H-pyrazoles via 3(5)-amino-4-(ethylsulfinyl)-1H-pyrazole desulfinylation

Frédéric Lassagne , Katia Snégaroff , Thierry Roisnel , Ekhlass Nassar , Florence Mongin et al.
Heterocyclic communications, 2011, 17, pp.139-145. ⟨10.1515/hc.2011.026⟩
Journal articles istex hal-00736464v1
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From simple quinoxalines to potent oxazolo[5,4-f]quinoxaline inhibitors of glycogen-synthase kinase 3 (GSK3)

Frédéric Lassagne , Camille Duguépéroux , Carlos Roca , Concepción Pérez , Ana Martínez et al.
Organic & Biomolecular Chemistry, 2020, 18 (1), pp.154-162. ⟨10.1039/C9OB02002K⟩
Journal articles hal-02396922v1
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Deproto-metallation and computed CH acidity of 2-aryl-1,2,3-triazoles.

Floris Chevallier , Thomas Blin , Elisabeth Nagaradja , Frédéric Lassagne , Thierry Roisnel et al.
Organic & Biomolecular Chemistry, 2012, 10 (25), pp.4878-85. ⟨10.1039/c2ob25554e⟩
Journal articles hal-01053777v1