|
|
cdc-like/dual-specificity tyrosine phosphorylation-regulated kinases inhibitor leucettine L41 induces mTOR-dependent autophagy: implication for Alzheimer's disease.
Xavier Fant
,
Emilie Durieu
,
Gaëtan Chicanne
,
Bernard Payrastre
,
Diego Sbrissa
et al.
Journal articles
inserm-01012086v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
An efficient approach to dispacamide A and its derivatives.
Solène Guihéneuf
,
Ludovic Paquin
,
François Carreaux
,
Emilie Durieu
,
Laurent Meijer
et al.
Journal articles
hal-00870469v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Structure-Activity Relationship in the Leucettine Family of Kinase Inhibitors
Tania Tahtouh
,
Emilie Durieu
,
Benoit Villiers
,
Celine Bruyere
,
Thu Lan Nguyen
et al.
Journal articles
hal-03512536v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Marine-Derived 2-Aminoimidazolone Alkaloids. Leucettamine B-Related Polyandrocarpamines Inhibit Mammalian and Protozoan DYRK & CLK Kinases
Nadège Loaëc
,
Eletta Attanasio
,
Benoît Villiers
,
Emilie Durieu
,
Tania Tahtouh
et al.
Journal articles
hal-01640115v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Synthesis of N,N'-bis(5-arylidene-4-oxo-3,5-dihydro-4H-imidazol-2-yl)diamines bearing various linkers and biological evaluation as potential inhibitors of kinases.
Wacothon Karime Coulibaly
,
Ludovic Paquin
,
Anoubilé Bénie
,
Yves-Alain Bekro
,
Emilie Durieu
et al.
Journal articles
istex
hal-00813182v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Microwave Assisted Organic Synthesis (MAOS) of New Dispacamide A Derivatives Bearing a Thiazolinone Platform, Biological Assays on Inhibition of Protein Kinases and Cell Effects
Solene Guiheneuf
,
Ludovic Paquin
,
Francois Carreaux
,
Emilie Durieu
,
Helene Benedetti
et al.
Journal articles
hal-01114583v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Selectivity, cocrystal structures, and neuroprotective properties of leucettines, a family of protein kinase inhibitors derived from the marine sponge alkaloid leucettamine B.
Tania Tahtouh
,
Jonathan M. Elkins
,
Panagis Filippakopoulos
,
Meera Soundararajan
,
Guillaume Burgy
et al.
Journal articles
hal-00870472v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
30th Franco-Belgian conference of pharmacochemistry
Charlotte Bouckaert
,
Eric Goffin
,
Sebastien Dilly
,
Julien Hanson
,
Lionel Pochet
et al.
Journal articles
hal-02141338v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Exploring the Synthesis of New 1-(4-Substitutedphenylamino) imidazo[1,5-a]indol-3-one Derivatives as Cyclized Analogs of Leucettines
Guillaume Burgy
,
Emmanuelle Limanton
,
François Carreaux
,
Emilie Durieu
,
Laurent Meijer
et al.
Journal articles
hal-01116022v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Chemical synthesis and biological validation of immobilized protein kinase inhibitory Leucettines.
Guillaume Burgy
,
Tania Tahtouh
,
Emilie Durieu
,
Béatrice Foll-Josselin
,
Emmanuelle Limanton
et al.
Journal articles
hal-00822733v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
New 5-ylidene rhodanine derivatives based on the dispacamide A model.
Solène Guihéneuf
,
Ludovic Paquin
,
François Carreaux
,
Emilie Durieu
,
Thierry Roisnel
et al.
Journal articles
hal-01017003v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|
|
|
Design and Microwave Synthesis of New (5Z) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5Z) 2-Amino-5-arylidene-1,3-thiazol-4(5H)-one as New Inhibitors of Protein Kinase DYRK1A
Khadidja Bourahla
,
Solène Guihéneuf
,
Emmanuelle Limanton
,
Ludovic Paquin
,
Rémy Le Guével
et al.
Journal articles
hal-03467664v1
|
Share
Gmail
Facebook
Twitter
LinkedIn
More
|