@article{bruel:hal-01086026, TITLE = {{Synthesis of new pyridazino[4,5-b]indol-4-ones and pyridazin-3(2H)-one analogs as DYRK1A inhibitors}}, AUTHOR = {Bruel, Am{\'e}lie and B{\'e}n{\'e}teau, Romain and Chabanne, Myl{\`e}ne and Lozach, Olivier and Le Guevel, R{\'e}my and Ravache, Myriam and B{\'e}n{\'e}detti, H{\'e}l{\`e}ne and Meijer, Laurent and Log{\'e}, C{\'e}dric and Robert, Jean-Michel}, URL = {https://univ-rennes.hal.science/hal-01086026}, JOURNAL = {{Bioorganic and Medicinal Chemistry Letters}}, PUBLISHER = {{Elsevier}}, VOLUME = {24}, NUMBER = {21}, PAGES = {5037 - 5040}, YEAR = {2014}, MONTH = Nov, DOI = {10.1016/j.bmcl.2014.09.017}, KEYWORDS = {4-Oxo-3 ; 4-dihydro-5H-pyridazino[4 ; 5-b]indole ; Pyridazin-3(2H)-one ; DYRK1A inhibitors ; Anti-proliferative effects ; Synthesis}, PDF = {https://univ-rennes.hal.science/hal-01086026/file/Synthesis%20of%20new%20pyridazino_accepted.pdf}, HAL_ID = {hal-01086026}, HAL_VERSION = {v1}, }